Publications 2015

- Vranic, B.Z., and Vandamme, T.F. (2015) Preliminary study of an offline simultaneous determination of metoprolol tartrate and hydrochlorothiazide in powders and tablets by reflectance near-infrared spectroscopy. Pharm. Dev. Technol. 20, 99-104.
- Vranic, B.Z., and Vandamme, T.F. (2015) Effect of simulated precompression, compression pressure and tableting speed on an offline diffuse transmittance and reflectance near-infrared spectral information of model intact caffeine tablets. Pharm. Dev. Technol. 20, 90-98.
- Vandamme, T.F. (2015) Rodent models for human diseases. Eur. J. Pharmacol. 759, 84-89.
- Khan, I.U., Stolch, L., Serra, C. A., Anton, N., Akasov, R., and Vandamme, T.F. (2015) Microfluidic conceived pH sensitive core-shell particles for dual drug delivery. Int. J. Pharm. 478, 78-87.
- Khan, I.U., Serra, C.A., Anton, N., and Vandamme, T.F. (2015) Production of nanoparticle drug delivery systems with microfluidics tools. Expert Opin. Drug Deliv. 12, 547-562.
- Khan, I.U., Serra, C.A., Anton, N., Er-Rafik, M., Blanck, C., Schmutz, M., Kraus, I., Messaddeq, N., Sutter, C., Anton, H., Klymchenko, A.S., and Vandamme, T.F. (2015) Microfluidic conceived Trojan microcarriers for oral delivery of nanoparticles. Int. J. Pharm. 493, 7-15.
- Diouf, L.A., Mbaye, G., Ndiaye, A., Sy, P.M., Djiboune, A.R., Soumboundou, M., Ndiaye, I.E., Anton, N., Vandamme, T.F., and Diarra, M. (2015) Peanut oil based W1/O/W2 multiple emulsions for oral administration of insulin. Int. J. Curr. Res. 7, 22420-22423.
- Neuberg, P., Périno, A., Morin-Picardat, E., Anton, N., Darwich, Z., Weltin, D., Mely, Y., Klymchenko, A. S., Remy, J.S., and Wagner, A. (2015) Photopolymerized micelles of diacetylene amphiphile : physical characterization and cell delivery properties. Chem. Comm. 51, 11595-11598.
- Attia, M.F., Anton, N., Bouchaala, R., Didier, P., Arntz, Y., Messaddeq, N., Klymchenko, A.S., Mely, Y., and Vandamme, T.F. (2015) Functionalization of nano-emulsions with an amino-silica shell at the oil-water interface. RSC Adv. 5, 74353-74361.
- Martinčič, R., Kuzmanovski, I., Wagner, A., and Novic, M. (2015) Development of models for prediction of the antioxidant activity of derivatives of natural compounds. Anal. Chem. Acta. 868, 23–35.
- Kolodych, S., Koniev, O., Baatarkhuu, Z., Bonnefoy, J.Y., Debaene, F., Cianferani, S., Van Dorsselaer, A., Wagner, A. (2015) CBTF : New amine-to-thiol coupling reagent for preparation of antibody conjugates with increased plasma stability. Bioconjugate Chem. 26,197-200.
- Jacques, S.A., Kuhn, I., Koniev, O., Schuber, F., Lund, F.E., Wagner, A., Muller-Steffner, H., and Kellenberger, E. (2015) Discovery of potent inhibitors of Schistosoma mansoni NAD+ catabolizing enzyme. J. Med. Chem. 8, 3582-92.
- Koniev, O., and Wagner, A. (2015) Developments and recent advancements in the field of endogenous amino acid selective bond forming reactions for bioconjugation. Chem. Soc. Rev. 44, 5495-5551.
- Neuberg, P., Périno, A., Morin-Picardat, E., Anton, N, Darwich, Z., Weltin, D. Mely, Y., Klymchenko, A.S., Remy, J.S., and Wagner, A. (2015) Photopolymerized micelles of diacetylene amphiphile : Physical characterization and cell delivery properties. Chem. Commun. 51, 11595-11598.
- Leriche, G., Jacques, S.A., Nothisen, M., Baumlin, N., Muller, C.D., Bagnard, D., Remy, J.S., Wagner, A. (2015) Spiro di-orthoester (SpiDo), a human plasma stable acid-sensitive cleavable linker for lysosomal release, Bioconjugate Chem. 26, 1461-1465.
- Koniev, O., Kolodych, S., Baatarkhuu, Z., Bonnefoy, J.Y., and Wagner, A. (2015) MAPN : New reagent for kinetically resolved thiol-to-thiol coupling. Bioconjugate Chem. 26, 1863−1867.
- Flacher, V., Neuberg, P., Point, F., Daubeuf, F., Muller, Q., Sigwalt, D., Fauny, J.D., Remy, J.S., Frossard, N., Wagner, A., Mueller, C.G., and Schaeffer, E.(2015) Mannoside glycolipid conjugates display antiinflammatory activity by inhibition of Toll-like Receptor-4 mediated cell activation. ACS Chem. Biol. 10, 2697-2705.
- Spanedda, M.V., Salome, C., Hilbold, B., Berner, E., Heurtault, B., Fournel, S., Frisch, B., and Bourel-Bonnet, L. (2015) Smart tools and orthogonal click-like reactions onto small unilamellar vesicles : Additional molecular data. Data in Brief 5, 145-154.
- Salome, C., Spanedda, M.V., Hilbold, B., Berner, E., Heurtault, B., Fournel, S., Frisch, B., and Bourel-Bonnet, L. (2015) Smart tools and orthogonal click-like reactions onto small unilamellar vesicles. Chem. Phys. Lipids 188, 27-36.
- Rios, C., Longo, J., Zahouani, S., Garnier, T., Vogt, C., Reisch, A., Senger, B., Boulmedais, F., Hemmerle, J., Benmlih, K., Frisch, B., Schaaf, P., Jierry, L., and Lavalle, P. (2015) A new biomimetic route to engineer enzymatically active mechano-responsive materials. Chem. Commun. 51, 5622-5.
- Kakhi, Z., Frisch, B., Bourel-Bonnet, L., Hemmerle, J., Pons, F., and Heurtault, B. (2015) Airway administration of a highly versatile peptide-based liposomal construct for local and distant antitumoral vaccination. Int. J. Pharm. 496, 1047-56.
- Pulka-Ziach, K., Pavet, V., Chekkat, N., Estieu-Gionnet, K., Rohac, R., Lechner, M. C., Smulski, C. R., Zeder-Lutz, G., Altschuh, D., Gronemeyer, H., Fournel, S., Odaert, B., and Guichard, G. (2015) Thioether analogues of disulfide-bridged cyclic peptides targeting death receptor 5 : conformational analysis, dimerisation and consequences for receptor activation. Chembiochem 16, 293-301.
- Pierrat, P., Wang, R., Kereselidze, D., Lux, M., Didier, P., Kichler, A., Pons, F., and Lebeau, L. (2015) Efficient in vitro and in vivo pulmonary delivery of nucleic acid by carbon dot-based nanocarriers. Biomaterials 51, 290-302.
- Kellenberger, S., and Grutter, T. (2015) Architectural and Functional Similarities between Trimeric ATP gated P2X receptors and acid-sensing ion channels. J. Mol. Biol. 427, 54-66.
- Habermacher, C., Dunning, K., Chataigneau, T., and Grutter, T. (2015) Molecular structure and function of P2X receptors. Neuropharmacol. 104, 18-30.
- Schmitt, J., Heitz, V., Sour, A., Bolze, F., Ftouni, H., Nicoud, J.F., Flamigni, L., and Ventura, B. (2015) Diketopyrrolopyrrole-porphyrin conjugates with high two-photon absorption and singlet oxygen generation for two-photon photodynamic therapy. Angew. Chem. Int. Ed. Engl. 54, 169-173.
- Guo, L., Chan, M.S., Xu, D., Tam, D.Y., Bolze, F., Lo, P.K., and Wong, M. S. (2015) Indole-based cyanine as a nuclear RNA-selective two-photon fluorescent probe for live cell imaging. ACS Chem. Biol. 10, 1171-1175.
- Dai, Z., Tam, D.Y., Xu, H., Chan, M.S., Liu, L.S., Bolze, F., Sun, X.H., and Lo, P.K. (2015) Conformational change of self-assembled DNA nanotubes induced by two-photon excitation. Small 11, 4090-4096.
- Chang, Y., Michelin, C., Bucher, L., Desbois, N., Gros, C.P., Piant, S., Bolze, F., Fang, Y., Jiang, X., and Kadish, K.M. (2015) Synthesis and characterization of carbazole-linked porphyrin tweezers. Chem.-Eur. J. 21, 12018-12025.
- Niehl, A. ; Appaix, F. ; Bosca, S., van der Sanden, B. ; Nicoud, J.F. ; Bolze, F., and Heinlein, M. (2015) Fluorescent tobacco mosaic virus-derived bio-nanoparticles for intravital two-photon imaging. Front. Plant Sci. 6, 1244.
- Douat, C., Aisenbrey, C., Antunes, S., Decossas, M., Lambert, O., Bechinger, B., Kichler, A., and Guichard, G. (2015) A cell-penetrating foldamer with a bioreducible linkage for intracellular delivery of DNA. Angew. Chem. Int. Ed. Engl. 54, 11133-7.
- Flacher, V., Neuberg, P., Point, F., Daubeuf, F., Muller, Q., Sigwalt, D., Fauny, J.D., Remy, J.S., Frossard, N., Wagner, A., Mueller, C.G., and Schaeffer, E. (2015) Mannoside glycolipid conjugates display antiinflammatory activity by inhibition of Toll-like Receptor-4 mediated cell activation. ACS Chem. Biol. 10, 2697-705.
- Orlov, I., Schertel, A., Zuber, G., Klaholz, B., Drillien, R., Weiss, E., Schultz, P., and Spehner, D. (2015) Live cell immunogold labelling of RNA polymerase II. Sci. Rep. 5, 8324.
- Ouahabi, A.A., Kotera, M., Charles, L., and Lutz, J.F. (2015) Synthesis of monodisperse sequence-coded polymers with chain lengths above DP100. ACS Macro Lett. 4, 1077-1080.
- Pierrat, P., and Lebeau, L. (2015) Characterization of titratable mmphiphiles in lipid membranes by fluorescence spectroscopy. Langmuir 31, 12362-12371.
- Pierrat, P., Wang, R., Kereselidze, D., Lux, M., Didier, P., Kichler, A., Pons, F., and Lebeau, L. (2015) Efficient in vitro and in vivo pulmonary delivery of nucleic acid by carbon dot-based nanocarriers. Biomaterials 51, 290-302.
- Postupalenko, V., Desplancq, D., Orlov, I., Arntz, Y., Spehner, D., Mely, Y., Klaholz, B. P., Schultz, P., Weiss, E., and Zuber, G. (2015) Protein delivery system containing a nickel-immobilized polymer for multimerization of affinity-purified His-tagged proteins enhances cytosolic transfer. Angew. Chem. Int. Ed. Engl. 54, 10583-10586.
- Yan, W., Seifermann, S. M., Pierrat, P., and Braese, S. (2015) Synthesis of highly functionalized C-60 fullerene derivatives and their applications in material and life sciences. Org. Biomol.Chem. 13, 25-54.
- Neuberg, P., Périno, A., Morin-Picardat, E., Anton, N, Darwich, Z., Weltin, D. Mely, Y., Klymchenko, A.S., Remy, J.S., Wagner, A. (2015) Photopolymerized micelles of diacetylene amphiphile : Physical characterization and cell delivery properties. Chem. Commun. 51, 11595-11598.
- Leriche, G., Jacques, S.A., Nothisen, M., Baumlin, N., Muller, C.D., Bagnard, D., Remy, J.S., Wagner, A. (2015) Spiro di-orthoester (SpiDo), a human plasma stable acid-sensitive cleavable linker for lysosomal release, Bioconjugate Chem. 26, 1461-1465.